2022 OCTOBER
Nucl Med Biol. 2022;114-115:49-57. N-(4-[18F]fluorobenzyl)cholylglycine, a potential tracer for positron emission tomography of enterohepatic circulation and drug-induced inhibition of ileal bile acid transport. A proof-of-concept PET/CT study in pigs. Frisch K, Mortensen FV, Munk OL, Gormsen LC, Alstrup AKO. PubMed
Drug Metab Pharmacokinet. 2022;46:100464. Comparison of the inhibitory properties of the fruit component naringenin and its glycosides against OATP1A2 genetic variants. Araki N, Morita T, Akiyoshi T, Kataoka H, Yajima K, Katayama K, Imaoka A, Ohtani H. PubMed
Basic Clin Pharmacol Toxicol. 2022;131:311-324. Drug metabolism and drug transport of the 100 most prescribed oral drugs. Ditte B Iversen, Nanna Elman Andersen, Ann-Cathrine Dalgård Dunvald , Anton Pottegård , Tore B Stage. PubMed
Clin Pharmacol Ther. 2022;In press. PharmVar GeneFocus: SLCO1B1. Ramsey LB, Gong L, Lee SB, Wagner JB, Zhou X, Sangkuhl K, Adams SM, Straka RJ, Empey PE, Boone EC, Klein TE, Niemi M, Gaedigk A. PubMed
Clin Pharmacol Ther. 2022;112:1098-1107. Organic Anion Transporter Gene variants associated with plasma exposure and long-term response to Atrasentan in patients with Diabetic Kidney Disease. Smeijer JD, Koomen JV, Kohan DE, McMurray JJV, Bakris GL, Correa-Rotter R, Hou FF, Kitzman DW, Makino H, Mayer G, Nowicki M, Perkovic V, Rossing P, Tobe S, Parving HH, de Zeeuw D, Heerspink HJL. PubMed
Int J Mol Sci. 2022;23:8457. Free cholesterol affects the function and localization of human Na+/Taurocholate Cotransporting Polypeptide (NTCP) and Organic Cation Transporter 1 (OCT1). Idowu JY, Hagenbuch B. PubMed
Front Physiol. 2022;13:969363. Using a competitive counterflow assay to identify novel cationic substrates of OATP1B1 and OATP1B3. Schnegelberger RD, Steiert B, Sandoval PJ, Hagenbuch B. PubMed
Int J Mol Sci. 2022;23:10177. In vitro characterization of renal drug transporter activity in kidney cancer. Caetano-Pinto P, Justian N, Dib M, Fischer J, Somova M, Burchardt M, Wolff I. PubMed
Int J Mol Sci. 2022;23:10758. In vitro rescue of the bile acid transport function of ABCB11 variants by CFTR potentiators. Mareux E, Lapalus M, Ben Saad A, Zelli R, Lakli M, Riahi Y, Almes M, Banet M, Callebaut I, Decout JL, Falguières T, Jacquemin E, Gonzales E. PubMed
Cell Res. 2022;32:773-776. Structure of human NTCP reveals the basis of recognition and sodium-driven transport of bile salts into the liver. Liu H, Irobalieva RN, Bang-Sørensen R, Nosol K, Mukherjee S, Agrawal P, Stieger B, Kossiakoff AA, Locher KP. PubMed